Brief Information of the Cell Line and Protein
Cell Line ID: CL000005 , TE 671
Synonyms
TE-671
TE671
TE671/RD
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_1756
Protein ID: PT03766 , Acetylcholine receptor subunit alpha
Gene Name CHRNA1
Organism Homo sapiens, Human
Protein Classification Ion channel
Uniprot ID P02708
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000005  Protein ID: PT03766
 
Compound ID Compound Name Compound Formula
CP0000212
()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane
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C11H13ClN2
 1
1
IC50 = 160 nM
   TI
   LI
   LO
   TS
CP0010311
5-[(1R,6R)-9-azabicyclo[4.2.1]non-2-en-2-yl]-3-ethyl-1,2-oxazole
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C13H18N2O
 1
1
IC50 = 4200 nM
   TI
   LI
   LO
   TS
CP0010369
5-[(1R,6R)-9-azabicyclo[4.2.1]non-2-en-2-yl]-3-propan-2-yl-1,2-oxazole
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C14H20N2O
 1
1
IC50 = 5500 nM
   TI
   LI
   LO
   TS
CP0021868
descyanothiacloprid
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C9H10ClN3S
 1
1
IC50 = 6000 nM
   TI
   LI
   LO
   TS
CP0009981
5-[(1R,6R)-9-azabicyclo[4.2.1]non-2-en-2-yl]-3-phenyl-1,2-oxazole
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C17H18N2O
 1
1
IC50 = 7800 nM
   TI
   LI
   LO
   TS
CP0009799
3-(6-Chloro-pyridin-3-ylmethyl)-3H-thiazol-(2E)-ylideneamine
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C9H8ClN3S
 1
1
IC50 = 8000 nM
   TI
   LI
   LO
   TS
CP0006324
(1R,2S,6R)-2-(3-methyl-1,2-oxazol-5-yl)-9-azabicyclo[4.2.1]nonan-2-ol
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C12H18N2O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0006816
(1R,2R,6R)-2-(3-methyl-1,2-oxazol-5-yl)-9-azabicyclo[4.2.1]nonan-2-ol
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C12H18N2O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0007629
(1R,9S)-3-methyl-5-oxa-4,12-diazatricyclo[7.2.1.02,6]dodeca-2(6),3-diene
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C10H14N2O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0007633
ethyl 5-[(1R,6R)-9-azabicyclo[4.2.1]non-2-en-2-yl]-1,2-oxazole-3-carboxylate
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C14H18N2O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0010370
ethyl (1R,9S)-5-oxa-4,12-diazatricyclo[7.2.1.02,6]dodeca-2(6),3-diene-3-carboxylate
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C12H16N2O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0009782
1-(6-Chloro-pyridin-3-ylmethyl)-imidazolidin-(2Z)-ylideneamine
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C9H11ClN4
 1
1
IC50 = 11000 nM
   TI
   LI
   LO
   TS
CP0000063
CAS_29790-52-1
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C10H14N2
 1
1
IC50 = 21000 nM
   TI
   LI
   LO
   TS
CP0244746
(2Z)-1-[(6-chloropyridin-3-yl)methyl]-2-(nitromethylidene)-1,3-diazinane
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C11H13ClN4O2
 1
1
IC50 = 81000 nM
   TI
   LI
   LO
   TS