Compound ID |
Compound Name |
Compound Formula |
CP0497804
|
4-methyl-1-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-ylpiperidine-4-carboxylic acid
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|
C26H31NO2
|
1
|
1 |
Ki = 3.162 nM
|
|
|
CP0493859
|
3-methyl-1-[(3S)-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-yl]pyrrolidine-3-carboxylic acid
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|
C25H29NO2
|
1
|
1 |
Ki = 10 nM
|
|
|
CP0374587
|
3-[4-(1,2-dimethyl-10H-imidazo[1,2-b][2]benzazepin-4-yl)piperazin-1-yl]-2,2-dimethylpropanoic acid
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|
C23H30N4O2
|
1
|
1 |
Ki = 15.85 nM
|
|
|
CP0472908
|
(3S)-N,N-dimethylspiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-amine
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|
C21H25N
|
1
|
1 |
Ki = 15.85 nM
|
|
|
CP0374588
|
3-[4-(1-chloro-10H-imidazo[1,2-b][2]benzazepin-4-yl)piperazin-1-yl]-2,2-dimethylpropanoic acid
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|
C21H25ClN4O2
|
1
|
1 |
Ki = 25.12 nM
|
|
|
CP0040455
|
(Z)-2-butenedioate;10-(1-methyl-4-piperidinylidene)-5H-benzo[1,2]cyclohepta[3,4-b]thiophen-4-one
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|
C19H19NOS
|
1
|
1 |
Ki = 31.62 nM
|
|
|
CP0497806
|
2-(1-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-ylazetidin-3-yl)acetic acid
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|
C24H27NO2
|
1
|
1 |
Ki = 39.81 nM
|
|
|
CP0477585
|
2,2-dimethyl-3-[4-(2-methyl-10H-imidazo[1,2-b][2]benzazepin-4-yl)piperazin-1-yl]propanoic acid
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|
C22H28N4O2
|
1
|
1 |
Ki = 63.1 nM
|
|
|
CP0279245
|
1-((1S)-5',11'-Dihydrospiro[cyclopentane-1,10'-dibenzo[a,d]-cyclohepten]-3-yl)-3-azetidinecarboxylic Acid
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|
C23H25NO2
|
1
|
1 |
Ki = 79.43 nM
|
|
|
CP0402437
|
3-[4-(2-chloro-10H-imidazo[1,2-b][2]benzazepin-4-yl)piperazin-1-yl]-2,2-dimethylpropanoic acid
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|
C21H25ClN4O2
|
1
|
1 |
Ki = 100 nM
|
|
|
CP0497802
|
1-[(3S)-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-yl]pyrrolidine-3-carboxylic acid
Show/Hide
|
C24H27NO2
|
1
|
1 |
Ki = 100 nM
|
|
|
CP0477603
|
3-[4-(1-methoxy-10H-imidazo[1,2-b][2]benzazepin-4-yl)piperazin-1-yl]-2,2-dimethylpropanoic acid
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|
C22H28N4O3
|
1
|
1 |
Ki = 158.49 nM
|
|
|
CP0340560
|
(-)-1-((1S)-5',11'-Dihydrospiro[cyclopentane-1,10'-dibenzo-[a,d]cyclohepten]-3-yl)-4-piperidinecarboxylic Acid
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|
C25H29NO2
|
1
|
1 |
Ki = 158.49 nM
|
|
|
CP0379543
|
4-hydroxy-1-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-ylpiperidine-4-carboxylic acid
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|
C25H29NO3
|
1
|
1 |
Ki = 251.19 nM
|
|
|
CP0523799
|
2-(1-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-ylazetidin-3-ylidene)acetic acid
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|
C24H25NO2
|
1
|
1 |
Ki = 251.19 nM
|
|
|
CP0374581
|
4-piperazin-1-yl-10H-imidazo[1,2-b][2]benzazepine
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|
C16H18N4
|
1
|
1 |
Ki = 316.23 nM
|
|
|
CP0374589
|
3-[4-(2-fluoro-10H-imidazo[1,2-b][2]benzazepin-4-yl)piperazin-1-yl]-2,2-dimethylpropanoic acid
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|
C21H25FN4O2
|
1
|
1 |
Ki = 316.23 nM
|
|
|
CP0342216
|
3-((1S)-5',11'-Dihydrospiro[cyclopentane-1,10'-dibenzo[a,d]-cyclohepten]-3-yl)-3-azabicyclo[3.1.0]hexane-1-carboxylic Acid
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|
C25H27NO2
|
1
|
1 |
Ki = 398.11 nM
|
|
|
CP0487906
|
3-[4-(10H-imidazo[1,2-b][2]benzazepin-4-yl)-2,6-dimethylpiperazin-1-yl]propanoic acid
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|
C21H26N4O2
|
1
|
1 |
Ki = 630.96 nM
|
|
|
CP0335817
|
1-(11'H-Spiro[cyclopentane-1,10'-dibenzo[b,f]oxepin]-3-yl)-3-azetidinecarboxylic Acid
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|
C22H23NO3
|
1
|
1 |
Ki = 794.33 nM
|
|
|
CP0379547
|
2-[1-[(3S)-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-yl]pyrrolidin-3-yl]acetic acid
Show/Hide
|
C25H29NO2
|
1
|
1 |
Ki = 1000 nM
|
|
|
CP0524075
|
2-(1-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-ylpiperidin-4-yl)acetic acid
Show/Hide
|
C26H31NO2
|
1
|
1 |
Ki = 1000 nM
|
|
|
CP0075436
|
(2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-ethyl]-piperidin-4-yl}-methanol
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|
C22H28FNO3
|
1
|
1 |
Ki = 1258.93 nM
|
|
|
CP0475730
|
(3R)-1-[(3S)-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-yl]piperidine-3-carboxylic acid
Show/Hide
|
C25H29NO2
|
1
|
1 |
Ki = 1258.93 nM
|
|
|
CP0497808
|
methyl 1-[(3S)-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-yl]-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C26H29NO2
|
1
|
1 |
Ki = 1258.93 nM
|
|
|
CP0505536
|
4-[(3S)-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-yl]piperazine-2-carboxylic acid
Show/Hide
|
C24H28N2O2
|
1
|
1 |
Ki = 1258.93 nM
|
|
|
CP0470855
|
3-[4-(10H-imidazo[1,2-b][2]benzazepin-4-yl)piperazin-1-yl]-2,2-dimethylpropanoic acid
Show/Hide
|
C21H26N4O2
|
1
|
1 |
Ki = 1584.89 nM
|
|
|
CP0493852
|
1-spiro[6H-benzo[b][1]benzoxepine-5,3'-cyclopentane]-1'-ylpiperidine-4-carboxylic acid
Show/Hide
|
C24H27NO3
|
1
|
1 |
Ki = 1584.89 nM
|
|
|
CP0374582
|
3-[4-(10H-imidazo[1,2-b][2]benzazepin-4-yl)piperazin-1-yl]propanoic acid
Show/Hide
|
C19H22N4O2
|
1
|
1 |
Ki > 794.33 nM
|
|
|
CP0374584
|
2-[[4-(10H-imidazo[1,2-b][2]benzazepin-4-yl)piperazin-1-yl]methyl]prop-2-enoic acid
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|
C20H22N4O2
|
1
|
1 |
Ki > 794.33 nM
|
|
|
CP0374585
|
3-[4-(10H-imidazo[1,2-b][2]benzazepin-4-yl)piperazin-1-yl]cyclobutane-1-carboxylic acid
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|
C21H24N4O2
|
1
|
1 |
Ki > 794.33 nM
|
|
|
CP0374583
|
3-[4-(10H-imidazo[1,2-b][2]benzazepin-4-yl)-1,4-diazepan-1-yl]-2,2-dimethylpropanoic acid
Show/Hide
|
C22H28N4O2
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0279246
|
3-[[(3R)-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-yl]amino]propanoic acid
Show/Hide
|
C22H25NO2
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0279247
|
3-[[(3S)-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-yl]amino]propanoic acid
Show/Hide
|
C22H25NO2
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0351011
|
1-((1S)-5',11'-Dihydrospiro[cyclopentane-1,10'-dibenzo[a,d]-cyclohepten]-3-yl)-1,2,5,6-tetrahydro-3-pyridinecarboxylic Acid
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|
C25H27NO2
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0379554
|
3-fluoro-1-[(3S)-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-yl]piperidine-3-carboxylic acid
Show/Hide
|
C25H28FNO2
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0379562
|
1-[(3R)-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-yl]-3,6-dihydro-2H-pyridine-5-carboxylic acid
Show/Hide
|
C25H27NO2
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0406094
|
1-(3-chloro-5-oxospiro[benzo[b][1]benzoxepine-6,3'-cyclopentane]-1'-yl)piperidine-4-carboxylic acid
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|
C24H24ClNO4
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0406107
|
1-spiro[6H-benzo[b][1]benzoxepine-5,3'-cyclopentane]-1'-yl-3,6-dihydro-2H-pyridine-5-carboxylic acid
Show/Hide
|
C24H25NO3
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0454555
|
4-fluoro-1-spiro[6H-benzo[b][1]benzoxepine-5,3'-cyclopentane]-1'-ylpiperidine-4-carboxylic acid
Show/Hide
|
C24H26FNO3
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0472909
|
1-(3-fluoro-5-oxospiro[benzo[b][1]benzothiepine-6,3'-cyclopentane]-1'-yl)piperidine-4-carboxylic acid
Show/Hide
|
C24H24FNO3S
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0493850
|
1-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-yl-3,6-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
|
C25H27NO2
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0493851
|
1-(6'-fluorospiro[cyclopentane-3,10'-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaene]-1-yl)-3,6-dihydro-2H-pyridine-5-carboxylic acid
Show/Hide
|
C25H26FNO2
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0493856
|
1-((1S)-5',11'-Dihydrospiro[cyclopentane-1,10'-dibenzo[a,d]-cyclohepten]-3-yl)-4-fluoro-4-piperidinecarboxylic Acid
Show/Hide
|
C25H28FNO2
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0497801
|
(3R)-1-(3-chloro-5-oxospiro[benzo[b][1]benzoxepine-6,3'-cyclopentane]-1'-yl)piperidine-3-carboxylic acid
Show/Hide
|
C24H24ClNO4
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0497803
|
4-[(3S)-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-yl]morpholine-2-carboxylic acid
Show/Hide
|
C24H27NO3
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0505534
|
1-spiro[6H-benzo[b][1]benzoxepine-5,3'-cyclopentane]-1'-yl-3,6-dihydro-2H-pyridine-4-carboxylic acid
Show/Hide
|
C24H25NO3
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0505545
|
(3R)-1-spiro[6H-benzo[b][1]benzoxepine-5,3'-cyclopentane]-1'-ylpiperidine-3-carboxylic acid
Show/Hide
|
C24H27NO3
|
1
|
1 |
Ki > 1995.26 nM
|
|
|
CP0511822
|
(1S,5R)-3-spiro[cyclopentane-3,9'-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaene]-1-yl-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
Show/Hide
|
C25H27NO2
|
1
|
1 |
Ki > 1995.26 nM
|
|
|