| Compound ID |
Compound Name |
Compound Formula |
|
CP0566455
|
US10668051, Compound Example 67
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|
C19H14F4N4O
|
1
|
| 1 |
IC50 = 20.37 nM
|
|
|
|
CP0535573
|
US10668051, Compound Example 84
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|
C18H14F4N4O2
|
1
|
| 1 |
IC50 = 20.79 nM
|
|
|
|
CP0446246
|
US10668051, Compound Example 104
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|
C20H17F3N4O
|
1
|
| 1 |
IC50 = 22.96 nM
|
|
|
|
CP0499841
|
US10668051, Compound Example 87
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|
C20H13F6N3O
|
1
|
| 1 |
IC50 = 32.59 nM
|
|
|
|
CP0529321
|
US10668051, Compound Example 78
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|
C18H15F3N4OS
|
1
|
| 1 |
IC50 = 34.11 nM
|
|
|
|
CP0535572
|
US10668051, Compound Example 82
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|
C17H13F4N5OS
|
1
|
| 1 |
IC50 = 35.72 nM
|
|
|
|
CP0453982
|
US10668051, Compound Example 7
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|
C23H23N3O
|
1
|
| 1 |
IC50 = 36.35 nM
|
|
|
|
CP0560554
|
US10668051, Compound Example 114
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|
C18H13F4N5O
|
1
|
| 1 |
IC50 = 37.58 nM
|
|
|
|
CP0488297
|
US10668051, Compound Example 111
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|
C18H14F3N5O
|
1
|
| 1 |
IC50 = 47.21 nM
|
|
|
|
CP0529320
|
US10668051, Compound Example 74
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|
C18H17F3N4S
|
1
|
| 1 |
IC50 = 48.02 nM
|
|
|
|
CP0529322
|
US10668051, Compound Example 83
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|
C18H14F4N4OS
|
1
|
| 1 |
IC50 = 48.17 nM
|
|
|
|
CP0549952
|
US10668051, Compound Example 72
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|
C20H17F3N4O
|
1
|
| 1 |
IC50 = 48.22 nM
|
|
|
|
CP0480740
|
US10668051, Compound Example 108
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|
C19H13F5N4O
|
1
|
| 1 |
IC50 = 50.58 nM
|
|
|
|
CP0535576
|
US10668051, Compound Example 126
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|
C16H11F5N4OS
|
1
|
| 1 |
IC50 = 52.62 nM
|
|
|
|
CP0529323
|
US10668051, Compound Example 106
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|
C19H14F4N4O
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0506850
|
US10668051, Compound Example 28
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|
C19H18FN5OS
|
1
|
| 1 |
IC50 = 60.31 nM
|
|
|
|
CP0457044
|
US10668051, Compound Example 1
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|
C19H19N5OS
|
1
|
| 1 |
IC50 = 62.44 nM
|
|
|
|
CP0515686
|
US10668051, Compound Example 113
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|
C18H14F3N5O
|
1
|
| 1 |
IC50 = 62.56 nM
|
|
|
|
CP0508994
|
US10668051, Compound Example 56
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|
C18H15F3N4O2
|
1
|
| 1 |
IC50 = 63.17 nM
|
|
|
|
CP0549970
|
US10668051, Compound Example 49
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|
C19H13Cl2F3N4O
|
1
|
| 1 |
IC50 = 65.49 nM
|
|
|
|
CP0446247
|
US10668051, Compound Example 107
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|
C19H13F5N4O
|
1
|
| 1 |
IC50 = 70.32 nM
|
|
|
|
CP0506852
|
US10668051, Compound Example 53
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|
C18H15F3N4OS
|
1
|
| 1 |
IC50 = 72.03 nM
|
|
|
|
CP0512891
|
US10668051, Compound Example 122
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|
C19H13F5N4O
|
1
|
| 1 |
IC50 = 72.11 nM
|
|
|
|
CP0566457
|
US10668051, Compound Example 93
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|
C19H15F4N5O
|
1
|
| 1 |
IC50 = 81.25 nM
|
|
|
|
CP0535574
|
US10668051, Compound Example 88
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|
C20H13F6N3O
|
1
|
| 1 |
IC50 = 98.58 nM
|
|
|
|
CP0443002
|
US10668051, Compound Example 100
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|
C20H13F6N3O
|
1
|
| 1 |
IC50 = 99.71 nM
|
|
|
|
CP0560669
|
US10668051, Compound Example 60
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|
C21H18F3N3O
|
1
|
| 1 |
IC50 = 119.7 nM
|
|
|
|
CP0549953
|
US10668051, Compound Example 79
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|
C20H14F5N3O
|
1
|
| 1 |
IC50 = 123.8 nM
|
|
|
|
CP0506853
|
US10668051, Compound Example 57
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|
C19H17F3N4O2
|
1
|
| 1 |
IC50 = 124.5 nM
|
|
|
|
CP0535570
|
US10668051, Compound Example 17
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|
C21H18Cl2N4O
|
1
|
| 1 |
IC50 = 129.6 nM
|
|
|
|
CP0529318
|
US10668051, Compound Example 15
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|
C21H20N4O
|
1
|
| 1 |
IC50 = 141.3 nM
|
|
|
|
CP0566454
|
US10668051, Compound Example 33
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|
C22H18F3N3O
|
1
|
| 1 |
IC50 = 145.1 nM
|
|
|
|
CP0566456
|
US10668051, Compound Example 86
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|
C21H17F4N3O
|
1
|
| 1 |
IC50 = 147.2 nM
|
|
|
|
CP0515685
|
US10668051, Compound Example 101
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|
C16H13F3N6OS
|
1
|
| 1 |
IC50 = 149.6 nM
|
|
|
|
CP0549847
|
US10668051, Compound Example 91
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|
C19H13F5N4O
|
1
|
| 1 |
IC50 = 159.1 nM
|
|
|
|
CP0549849
|
US10668051, Compound Example 92
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|
C19H12Cl2F4N4O
|
1
|
| 1 |
IC50 = 159.3 nM
|
|
|
|
CP0535571
|
US10668051, Compound Example 37
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|
C19H17ClFN5OS
|
1
|
| 1 |
IC50 = 181.1 nM
|
|
|
|
CP0529319
|
US10668051, Compound Example 52
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|
C17H14F3N5OS
|
1
|
| 1 |
IC50 = 183.6 nM
|
|
|
|
CP0549939
|
US10668051, Compound Example 35
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|
C21H19FN4O
|
1
|
| 1 |
IC50 = 184.6 nM
|
|
|
|
CP0499840
|
US10668051, Compound Example 80
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|
C18H14ClF3N4OS
|
1
|
| 1 |
IC50 = 194 nM
|
|
|
|
CP0560552
|
US10668051, Compound Example 89
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|
C19H14F4N4O
|
1
|
| 1 |
IC50 = 205.7 nM
|
|
|
|
CP0441591
|
US10668051, Compound Example 2
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|
C20H20N4OS
|
1
|
| 1 |
IC50 = 206.7 nM
|
|
|
|
CP0453983
|
US10668051, Compound Example 36
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|
C21H20FN5O
|
1
|
| 1 |
IC50 = 223.5 nM
|
|
|
|
CP0516943
|
US10668051, Compound Example 90
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|
C19H14F4N4O
|
1
|
| 1 |
IC50 = 232 nM
|
|
|
|
CP0535569
|
US10668051, Compound Example 16
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|
C21H19FN4O
|
1
|
| 1 |
IC50 = 243.9 nM
|
|
|
|
CP0560670
|
US10668051, Compound Example 66
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|
C19H15F3N4O
|
1
|
| 1 |
IC50 = 254.7 nM
|
|
|
|
CP0549938
|
US10668051, Compound Example 4
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|
C20H20N4O2
|
1
|
| 1 |
IC50 = 256.1 nM
|
|
|
|
CP0560551
|
US10668051, Compound Example 76
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|
C18H16F3N5OS
|
1
|
| 1 |
IC50 = 269 nM
|
|
|
|
CP0488299
|
US10668051, Compound Example 124
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|
C18H12F5N5O
|
1
|
| 1 |
IC50 = 295.4 nM
|
|
|
|
CP0535575
|
US10668051, Compound Example 125
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|
C16H12F4N4OS
|
1
|
| 1 |
IC50 = 373.4 nM
|
|
|
|
CP0549940
|
US8921364, 45
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|
C21H18F2N4O
|
1
|
| 1 |
IC50 = 436.1 nM
|
|
|
|
CP0575687
|
US10668051, Compound Example 19
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|
C23H23N3O
|
1
|
| 1 |
IC50 = 456.6 nM
|
|
|
|
CP0560553
|
US10668051, Compound Example 97
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|
C19H16F4N6O
|
1
|
| 1 |
IC50 = 600.3 nM
|
|
|
|
CP0457045
|
US10668051, Compound Example 71
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|
C20H17F3N4O
|
1
|
| 1 |
IC50 = 604.3 nM
|
|
|
|
CP0506851
|
BDBM444852
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|
C20H21N5OS
|
1
|
| 1 |
IC50 = 851.4 nM
|
|
|
|
CP0512900
|
US10668051, Compound Example 22
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|
C22H22N4O
|
1
|
| 1 |
IC50 = 968.1 nM
|
|
|
