| Compound ID |
Compound Name |
Compound Formula |
|
CP0852693
|
(R)-2-(2-methyl-4-((3-(2-oxo-3,4-dihydro-2H-benzo[e][1,3]oxazin-6-yl)-1H-pyrazol-4-yl)methyl)piperazin-1-yl)isonicotinonitrile
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C23H23N7O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0859383
|
6-(4-((2-(trifluoromethyl)-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
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C23H20F6N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0859900
|
(S)-6-(4-((2-(hydroxymethyl)-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
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|
C23H23F3N6O3
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0859901
|
(S)-6-(4-((2-(fluoromethyl)-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
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|
C23H22F4N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0861970
|
(S)-6-(4-((3-(fluoromethyl)-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
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|
C23H22F4N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0861971
|
(S)-1-((3-(2-oxo-3,4-dihydro-2H-benzo[e][1,3]oxazin-6-yl)-1H-pyrazol-4-yl)methyl)-4-(5-(trifluoromethyl)pyridin-2-yl)piperazine-2-carboxylic acid
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|
C23H21F3N6O4
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0864750
|
(S)-6-(4-((3-methyl-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-2H-benzo[e][1,3]oxazine-2,4(3H)-dione
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|
C23H21F3N6O3
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0864751
|
(R)-7-(4-((3-methyl-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-1,2-dihydroisoquinolin-3(4H)-one
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|
C24H25F3N6O
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0864756
|
(R)-7-(4-((3-methyl-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)isoquinoline-1,3(2H,4H)-dione
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|
C24H23F3N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
|
CP0866493
|
(R)-6-(4-((3-methyl-4-(4-(trifluoromethyl)phenyl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C24H24F3N5O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
|
CP0866684
|
6-(4-((3-(trifluoromethyl)-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C23H20F6N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0866685
|
(S)-6-(4-((3-methyl-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)benzo[d]oxazol-2(3H)-one
Show/Hide
|
C22H21F3N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
|
CP0867178
|
6-(4-((4-(5-(trifluoromethyl)pyridin-2-yl)-1,4-diazepan-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydroquinazolin-2(1H)-one
Show/Hide
|
C23H24F3N7O
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
|
CP0867179
|
(R)-6-(5-((3-methyl-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-2H-1,2,3-triazol-4-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C22H22F3N7O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
|
CP0867180
|
6-(4-((4-(5-(trifluoromethyl)pyridin-2-yl)-4,7-diazaspiro[2.5]octan-7-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C24H23F3N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
|
CP0876655
|
6-(4-((4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C22H21F3N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0895828
|
(R)-6-(4-((3-methyl-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)benzo[d]oxazol-2(3H)-one
Show/Hide
|
C22H21F3N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
|
CP0895829
|
6-(4-((3-(5-(trifluoromethyl)pyridin-2-yl)-3,6-diazabicyclo[3.1.1]heptan-6-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C23H21F3N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
|
CP0895830
|
6-(4-((4-(5-(trifluoromethyl)pyridin-2-yl)-1,4-diazepan-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C23H23F3N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
|
CP0903808
|
(S)-6-(4-((3-(hydroxymethyl)-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C23H23F3N6O3
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
|
CP0903809
|
(R)-6-(4-((3-methyl-4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C24H24F3N5O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
|
CP0921238
|
(R)-6-(4-((4-(2-fluorobenzyl)-3-methylpiperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C24H26FN5O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0921264
|
(R)-6-(4-((4-(4-chlorophenyl)-3-methylpiperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C23H24ClN5O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0934278
|
(R)-6-(4-((3-methyl-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-2H-benzo[e][1,3]oxazine-2,4(3H)-dione
Show/Hide
|
C23H21F3N6O3
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0934279
|
6-(4-((3-(5-(trifluoromethyl)pyridin-2-yl)-3,8-diazabicyclo[3.2.1]octan-8-yl)methyl)-1H-pyrazol-3-yl)-2H-benzo[e][1,3]oxazine-2,4(3H)-dione
Show/Hide
|
C24H21F3N6O3
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0934280
|
(S)-6-(4-((3-(trifluoromethyl)-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C23H20F6N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0934281
|
(R)-6-(2-methyl-4-((3-(2-oxo-3,4-dihydro-2H-benzo[e][1,3]oxazin-6-yl)-1H-pyrazol-4-yl)methyl)piperazin-1-yl)nicotinonitrile
Show/Hide
|
C23H23N7O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0935590
|
(R)-6-(4-((4-cyclohexyl-3-methylpiperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C23H31N5O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0935722
|
7-(4-((4-(5-(trifluoromethyl)pyridin-2-yl)-1,4-diazepan-1-yl)methyl)-1H-pyrazol-3-yl)-1,2-dihydroisoquinolin-3(4H)-one
Show/Hide
|
C24H25F3N6O
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0935723
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(R)-6-(4-((3-methyl-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydroquinazolin-2(1H)-one
Show/Hide
|
C23H24F3N7O
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0951006
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6-(4-((4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-2H-benzo[e][1,3]oxazine-2,4(3H)-dione
Show/Hide
|
C22H19F3N6O3
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0951007
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(R)-5-(4-((3-methyl-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)benzo[d]oxazol-2(3H)-one
Show/Hide
|
C22H21F3N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0951008
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6-(4-((4-(2,3-dimethylphenyl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-2H-benzo[e][1,3]oxazine-2,4(3H)-dione
Show/Hide
|
C24H25N5O3
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0951009
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(S)-6-(4-((3-methyl-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C23H23F3N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0952202
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(R)-6-(4-((3-methyl-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C23H23F3N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0952203
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6-(4-((3-(5-(trifluoromethyl)pyridin-2-yl)-3,8-diazabicyclo[3.2.1]octan-8-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C24H23F3N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0952204
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(R)-6-(4-((3-(trifluoromethyl)-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C23H20F6N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0952205
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(R)-6-(4-((3-methyl-4-(5-methylpyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C23H26N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0952214
|
(R)-6-(4-((3-methyl-4-(4-(trifluoromethyl)pyrimidin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C22H22F3N7O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0952215
|
(R)-4,4-dimethyl-6-(4-((3-methyl-4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C25H27F3N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0952860
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6-(4-((4-(2,3-dimethylphenyl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)benzo[d]oxazol-2(3H)-one
Show/Hide
|
C23H25N5O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0954845
|
6-(4-((4-(5-(trifluoromethyl)pyridin-2-yl)piperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[b][1,4]oxazin-2-one
Show/Hide
|
C22H21F3N6O2
|
1
|
| 1 |
IC50 < 500 nM
|
|
|
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CP0968100
|
(R)-6-(4-((4-(5-chloropyridin-2-yl)-3-methylpiperazin-1-yl)methyl)-1H-pyrazol-3-yl)-3,4-dihydro-2H-benzo[e][1,3]oxazin-2-one
Show/Hide
|
C22H23ClN6O2
|
1
|
| 1 |
IC50 < 500 nM
|
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