Brief Information of the Cell Line and Protein
Cell Line ID: CL000001 , Jurkat
Synonyms
JURKAT
JM
JM-Jurkat
Jurkat-FHCRC
Jurkat FHCRC
FHCRC-11
FHCRC subclone 11
FCCH1024
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0065
Protein ID: PT06229 , Calcium release-activated calcium channel protein 1
Gene Name ORAI1
Organism Homo sapiens, Human
Protein Classification Ion channel
Uniprot ID Q96D31
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000001  Protein ID: PT06229
 
Compound ID Compound Name Compound Formula
CP0563903
US8993612, 20
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C21H17F3N6O
 1
1
IC50 = 39.17 nM
   TI
   LI
   LO
   TS
CP0451908
US8993612, 6
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C23H22N6O
 1
1
IC50 = 51.31 nM
   TI
   LI
   LO
   TS
CP0550626
US8993612, 18
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C22H16F3N5O
 1
1
IC50 = 53.36 nM
   TI
   LI
   LO
   TS
CP0888321
US8993612, 17
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C23H17F3N4O
 1
1
IC50 = 86.12 nM
   TI
   LI
   LO
   TS
CP0451910
US8993612, 21
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C21H17F3N6O
 1
1
IC50 = 139 nM
   TI
   LI
   LO
   TS
CP0550232
US8993612, 10
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C26H24N4O
 1
1
IC50 = 146.7 nM
   TI
   LI
   LO
   TS
CP0563904
US8993612, 30
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C21H16F4N6O
 1
1
IC50 = 160.5 nM
   TI
   LI
   LO
   TS
CP0545628
US8993612, 2
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C22H20N6O
 1
1
IC50 = 182.5 nM
   TI
   LI
   LO
   TS
CP0556419
US8993612, 12
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C26H23FN4O
 1
1
IC50 = 263.2 nM
   TI
   LI
   LO
   TS
CP0559652
US8993612, 5
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C24H23N5O
 1
1
IC50 = 383.1 nM
   TI
   LI
   LO
   TS