| Compound ID |
Compound Name |
Compound Formula |
|
CP0149360
|
N-ethyl-4-[4-[(8-methoxy-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-3-methylbenzamide
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|
C25H32N4O4
|
2
|
| 1 |
EC50 = 10 nM
|
|
|
| 2 |
EC50 = 44000 nM
|
|
|
|
CP0294871
|
3-chloro-N-cyclopropyl-4-[4-[(2,8-dimethyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]benzamide
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|
C25H29ClN4O3
|
2
|
| 1 |
EC50 = 10 nM
|
|
|
| 2 |
EC50 = 43000 nM
|
|
|
|
CP0087307
|
4-[4-[(8-ethoxy-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-N,3-dimethylbenzamide
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|
C25H32N4O4
|
2
|
| 1 |
EC50 = 20 nM
|
|
|
| 2 |
EC50 = 26000 nM
|
|
|
|
CP0176396
|
N-cyclopropyl-4-[4-[(8-methoxy-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-3-methylbenzamide
Show/Hide
|
C26H32N4O4
|
2
|
| 1 |
EC50 = 20 nM
|
|
|
| 2 |
EC50 = 77000 nM
|
|
|
|
CP0351323
|
N-cyclopropyl-4-[4-[(8-ethoxy-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-3-methylbenzamide
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|
C27H34N4O4
|
2
|
| 1 |
EC50 = 20 nM
|
|
|
| 2 |
EC50 = 100000 nM
|
|
|
|
CP0351324
|
4-[4-[(8-ethoxy-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-N-ethyl-3-methylbenzamide
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|
C26H34N4O4
|
2
|
| 1 |
EC50 = 20 nM
|
|
|
| 2 |
EC50 = 100000 nM
|
|
|
|
CP0120515
|
4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbonyl]-4-fluorophenyl}methyl)-1,2-dihydrophthalazin-1-one
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|
C24H23FN4O3
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0286789
|
4-[4-[(8-methoxy-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-N,3-dimethylbenzamide
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|
C24H30N4O4
|
2
|
| 1 |
EC50 = 60 nM
|
|
|
| 2 |
EC50 = 100000 nM
|
|
|
|
CP0037604
|
(S)-2-(4-(piperidin-3-yl)phenyl)-2H-indazole-7-carboxamide
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|
C19H20N4O
|
2
|
| 1 |
EC50 = 200 nM
|
|
|
| 2 |
EC50 = 31000 nM
|
|
|
|
CP0044519
|
2-[(2R)-2-methylpyrrolidin-2-yl]-1H-1,3-benzodiazole-4-carboxamide
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|
C13H16N4O
|
1
|
| 1 |
EC50 = 3000 nM
|
|
|
|
CP0338396
|
3-chloro-N-ethyl-4-[4-[(2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]benzamide
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|
C23H27ClN4O3
|
2
|
| 1 |
EC50 = 4000 nM
|
|
|
| 2 |
EC50 = 100000 nM
|
|
|
|
CP0149364
|
N-cyclopropyl-4-[4-[(2,8-dimethyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]benzamide
Show/Hide
|
C25H30N4O3
|
2
|
| 1 |
EC50 = 5000 nM
|
|
|
| 2 |
EC50 = 100000 nM
|
|
|
|
CP0149362
|
4-[4-[(2,8-dimethyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-N-ethyl-3-methylbenzamide
Show/Hide
|
C25H32N4O3
|
2
|
| 1 |
EC50 = 9000 nM
|
|
|
| 2 |
EC50 = 55000 nM
|
|
|
|
CP0369505
|
4-[4-[(2,8-dimethyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-N,3-dimethylbenzamide
Show/Hide
|
C24H30N4O3
|
2
|
| 1 |
EC50 = 9000 nM
|
|
|
| 2 |
EC50 = 78000 nM
|
|
|
|
CP0429934
|
4-[4-[(2,8-dimethyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-N-ethylbenzamide
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|
C24H30N4O3
|
2
|
| 1 |
EC50 = 9000 nM
|
|
|
| 2 |
EC50 = 94000 nM
|
|
|
|
CP0149365
|
4-[4-[(2,8-dimethyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-N-methylbenzamide
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|
C23H28N4O3
|
2
|
| 1 |
EC50 = 11000 nM
|
|
|
| 2 |
EC50 = 75000 nM
|
|
|
|
CP0524813
|
N-methyl-4-[4-[(2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]benzamide
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|
C22H26N4O3
|
2
|
| 1 |
EC50 = 14000 nM
|
|
|
| 2 |
EC50 = 15000 nM
|
|
|
|
CP0176398
|
3-chloro-4-[4-[(2,8-dimethyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-N-methylbenzamide
Show/Hide
|
C23H27ClN4O3
|
2
|
| 1 |
EC50 = 14000 nM
|
|
|
| 2 |
EC50 = 45000 nM
|
|
|
|
CP0338049
|
3-chloro-4-[4-[(2,8-dimethyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-N-ethylbenzamide
Show/Hide
|
C24H29ClN4O3
|
2
|
| 1 |
EC50 = 14000 nM
|
|
|
| 2 |
EC50 = 47000 nM
|
|
|
|
CP0087309
|
N-ethyl-4-[4-[(2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]benzamide
Show/Hide
|
C23H28N4O3
|
2
|
| 1 |
EC50 = 15000 nM
|
|
|
| 2 |
EC50 = 42000 nM
|
|
|
|
CP0044521
|
N-cyclopropyl-4-[4-[(8-methoxy-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]benzamide
Show/Hide
|
C25H30N4O4
|
1
|
| 1 |
EC50 = 16000 nM
|
|
|
|
CP0087308
|
N-ethyl-4-[4-[(8-methoxy-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]benzamide
Show/Hide
|
C24H30N4O4
|
1
|
| 1 |
EC50 = 16000 nM
|
|
|
|
CP0351325
|
N-cyclopropyl-4-[4-[(2,8-dimethyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-3-methylbenzamide
Show/Hide
|
C26H32N4O3
|
2
|
| 1 |
EC50 = 18000 nM
|
|
|
| 2 |
EC50 = 100000 nM
|
|
|
|
CP0338050
|
4-[4-[(8-methoxy-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl)methyl]piperazin-1-yl]-N-methylbenzamide
Show/Hide
|
C23H28N4O4
|
1
|
| 1 |
EC50 = 27000 nM
|
|
|
