Brief Information of the Compound and Protein
Compound Name
 Compound Info 
5-[2-[(1S)-1-cyclopropylethyl]-7-methyl-1-oxo-3H-isoindol-5-yl]-N-(1-methylpyrazol-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
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 PubChem ID
CID: 168293104
Canonical SMILES
C[C@@H](C1CC1)N1Cc2cc(cc(C)c2C1=O)-c1ccn2ncc(C(=O)Nc3cnn(C)c3)c2n1
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Compound Formula C25H25N7O2
Compound Structure
Protein Name
 Protein Info 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Protein Classification
Enzyme
>
Transferase
Uniprot ID
P48736
Gene Name
PIK3CG
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000040 THP-1
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 638 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 34.1 nM