Brief Information of the Compound and Protein
Compound Name
2-[4-[4-[(2-oxo-3,4-dihydro-1H-quinolin-7-yl)oxy]butyl]piperazin-1-yl]pyridine-3-carbonitrile
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PubChem ID
CID: 168291109
Canonical SMILES
O=C1CCc2ccc(OCCCCN3CCN(CC3)c3ncccc3C#N)cc2N1
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Compound Formula C23H27N5O2
Compound Structure
Protein Name
5-hydroxytryptamine receptor 2A
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P28223
Gene Name
HTR2A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
Ki = 7400 nM
   TI
   LI
   LO
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