Brief Information of the Compound and Protein
Compound Name
2-[[7-(4-chloro-2,5-dioxopyrrol-3-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]oxy]-5-fluorobenzonitrile
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PubChem ID
CID: 168286083
Canonical SMILES
Fc1ccc(Oc2ncnc3CN(CCc23)C2=C(Cl)C(=O)NC2=O)c(c1)C#N
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Compound Formula C18H11ClFN5O3
Compound Structure
Protein Name
Short transient receptor potential channel 5
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9UL62
Gene Name
TRPC5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 664 nM
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