Brief Information of the Compound and Protein
Compound Name
3-chloro-4-[2-cyclopropyl-4-[4-fluoro-2-(trifluoromethyl)phenoxy]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]pyrrole-2,5-dione
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PubChem ID
CID: 168297837
Canonical SMILES
Fc1ccc(Oc2nc(nc3CN(CCc23)C2=C(Cl)C(=O)NC2=O)C2CC2)c(c1)C(F)(F)F
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Compound Formula C21H15ClF4N4O3
Compound Structure
Protein Name
Short transient receptor potential channel 5
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9UL62
Gene Name
TRPC5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 2080 nM
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