Brief Information of the Compound and Protein
Compound Name
3-chloro-4-[4-[2-(trifluoromethyl)phenoxy]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]pyrrole-2,5-dione
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PubChem ID
CID: 168293268
Canonical SMILES
FC(F)(F)c1ccccc1Oc1ncnc2CN(CCc12)C1=C(Cl)C(=O)NC1=O
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Compound Formula C18H12ClF3N4O3
Compound Structure
Protein Name
Short transient receptor potential channel 5
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9UL62
Gene Name
TRPC5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 452 nM
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