Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(3S)-N-[(3-chloro-2,4-difluorophenyl)-[5-chloro-6-(trifluoromethyl)pyridin-3-yl]methyl]-5-oxopyrrolidine-3-carboxamide
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Canonical SMILES
Fc1ccc(C(NC(=O)[C@@H]2CNC(=O)C2)c2cnc(c(Cl)c2)C(F)(F)F)c(F)c1Cl
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Compound Formula C18H12Cl2F5N3O2
Compound Structure
Protein Name
 Protein Info 
Sodium channel protein type 8 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q9UQD0
Gene Name
SCN8A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 4.2 nM
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