Brief Information of the Compound and Protein
Compound Name
4-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-N-(1H-indazol-6-yl)piperazine-1-carboxamide
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PubChem ID
CID: 168269878
Canonical SMILES
FC(F)(F)c1cnc(N2CCN(CC2)C(=O)Nc2ccc3cn[nH]c3c2)c(Cl)c1
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Compound Formula C18H16ClF3N6O
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 69 nM
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