Brief Information of the Compound and Protein
Compound Name
3-[2-(dimethylamino)ethyl]-1H-indol-4-ol
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PubChem ID
CID: 4980
SID: 15195604
Canonical SMILES
CN(C)CCc1c[nH]c2cccc(O)c12
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Compound Formula C12H16N2O
Compound Structure
Protein Name
5-hydroxytryptamine receptor 2A
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P28223
Gene Name
HTR2A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
IC50 = 8.34 nM
   TI
   LI
   LO
   TS
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 6.5 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 75.2 nM