Brief Information of the Compound and Protein
Compound Name
 Compound Info 
US9546164, 100
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 PubChem ID
CID: 118110531
Canonical SMILES
C[C@H](N1CCC(COc2cc(F)c(cc2C2CC2)C(=O)NS(C)(=O)=O)CC1)c1cc(Cl)cc(Cl)c1
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Compound Formula C25H29Cl2FN2O4S
Compound Structure
Protein Name
 Protein Info 
Sodium channel protein type 7 subunit alpha
Protein Classification
Ion channel
>
Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q01118
Gene Name
SCN7A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  3
1
IC50 = 0.6 nM
   TI
   LI
   LO
   TS
2
IC50 = 1.8 nM
   TI
   LI
   LO
   TS
3
IC50 = 16 nM
   TI
   LI
   LO
   TS