Brief Information of the Compound and Protein
Compound Name
 Compound Info 
N-(2-methyl-6-morpholin-4-ylpyridin-3-yl)-N-(2-methylpropyl)-2-(oxan-4-yl)-4-oxo-2,3-dihydrochromene-6-sulfonamide
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 PubChem ID
CID: 142380230
Canonical SMILES
CC(C)CN(c1ccc(nc1C)N1CCOCC1)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
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Compound Formula C28H37N3O6S
Compound Structure
Protein Name
 Protein Info 
Nuclear receptor ROR-gamma
Protein Classification
Transcription factor
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Nuclear receptor
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Nuclear hormone receptor subfamily 1
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Nuclear hormone receptor subfamily 1 group F
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Nuclear hormone receptor subfamily 1 group F member 3
Uniprot ID
P51449
Gene Name
RORC
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000001 Jurkat
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 19 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 8 nM