Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-[2-(4-chlorophenyl)ethyl]-1-[(E)-(7-ethyl-5-hydroxy-1H-indol-3-yl)methylideneamino]guanidine
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 PubChem ID
CID: 138319674
Canonical SMILES
CCc1cc(O)cc2c(\C=N\NC(=N)NCCc3ccc(Cl)cc3)c[nH]c12
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Compound Formula C20H22ClN5O
Compound Structure
Protein Name
 Protein Info 
Relaxin-3 receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Relaxin-like peptide receptor (family A GPCR)
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Relaxin receptor
Uniprot ID
Q9NSD7
Gene Name
RXFP3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  3
1
EC50 = 18.2 nM
   TI
   LI
   LO
   TS
2
EC50 = 22 nM
   TI
   LI
   LO
   TS
3
Ki = 274 nM
   TI
   LI
   LO
   TS