Brief Information of the Compound and Protein
Compound Name
3-amino-4-[4-[4-(dimethylamino)-4-oxobutyl]-2-fluorophenoxy]-6-methylthieno[2,3-b]pyridine-2-carboxamide
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PubChem ID
CID: 155515868
Canonical SMILES
CN(C)C(=O)CCCc1ccc(Oc2cc(C)nc3sc(C(N)=O)c(N)c23)c(F)c1
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Compound Formula C21H23FN4O3S
Compound Structure
Protein Name
Cyclin-dependent kinase 8
Protein Classification
Enzyme
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Kinase
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Protein Kinase
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CMGC protein kinase group
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CMGC protein kinase CDK family
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CMGC protein kinase CDK8 subfamily
Uniprot ID
P49336
Gene Name
CDK8
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 4.5 nM
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