Brief Information of the Compound and Protein
Compound Name
 Compound Info 
7-(4-methylsulfonylphenyl)-N-[2-(4-propan-2-yloxyphenyl)pyridin-4-yl]quinolin-4-amine
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Canonical SMILES
CC(C)Oc1ccc(cc1)-c1cc(Nc2ccnc3cc(ccc23)-c2ccc(cc2)S(C)(=O)=O)ccn1
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Compound Formula C30H27N3O3S
Compound Structure
Protein Name
 Protein Info 
TGF-beta receptor type-1
Protein Classification
Enzyme
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Kinase
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Protein Kinase
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TKL protein kinase group
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TKL protein kinase STKR family
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TKL protein kinase STKR Type 1 subfamily
Uniprot ID
P36897
Gene Name
TGFBR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 127.3 nM
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