Brief Information of the Compound and Protein
Compound Name
2-fluoro-6-[6-methyl-5-(5-methylthiophen-2-yl)-3-(2-phenylethyl)pyrazin-2-yl]phenol
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PubChem ID
CID: 135903265
SID: 57248669
Canonical SMILES
Cc1ccc(s1)-c1nc(CCc2ccccc2)c(nc1C)-c1cccc(F)c1O
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Compound Formula C24H21FN2OS
Compound Structure
Protein Name
Extracellular calcium-sensing receptor
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Ion receptor (family C GPCR)
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Calcium sensing receptor
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Calcium sensing receptor
Uniprot ID
P41180
Gene Name
CASR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 110 nM
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