Brief Information of the Compound and Protein
Compound Name
3-pyrazin-2-yl-N-[1-(trifluoromethyl)cyclobutyl]-11-oxa-3,4-diazatricyclo[6.2.1.02,6]undeca-2(6),4-diene-5-carboxamide
    Show/Hide
PubChem ID
CID: 156248679
Canonical SMILES
FC(F)(F)C1(CCC1)NC(=O)c1nn(c2C3CCC(Cc12)O3)-c1cnccn1
    Show/Hide
Compound Formula C18H18F3N5O2
Compound Structure
Protein Name
Cannabinoid receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Lipid-like ligand receptor (family A GPCR)
>
Cannabinoid receptor
Uniprot ID
P21554
Gene Name
CNR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 0.04 nM
   TI
   LI
   LO
   TS