Brief Information of the Compound and Protein
Compound Name
1-[[4-[(2-phenylacetyl)amino]pyrazol-1-yl]methyl]-N-[4-(trifluoromethyl)phenyl]pyrazole-3-carboxamide
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Canonical SMILES
FC(F)(F)c1ccc(NC(=O)c2ccn(Cn3cc(NC(=O)Cc4ccccc4)cn3)n2)cc1
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Compound Formula C23H19F3N6O2
Compound Structure
Protein Name
Hypoxia-inducible factor 1-alpha
Protein Classification
Transcription factor
Uniprot ID
Q16665
Gene Name
HIF1A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000017 HeLa Homo sapiens (Human)  1
1
IC50 = 1400 nM
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