Brief Information of the Compound and Protein
Compound Name
1-(2-oxo-1H-quinolin-5-yl)-3-[[2-(3-propan-2-ylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]methyl]urea
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Canonical SMILES
CC(C)c1cccc(c1)-n1nc(cc1CNC(=O)Nc1cccc2[nH]c(=O)ccc12)C(F)(F)F
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Compound Formula C24H22F3N5O2
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 0.88 nM
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