Brief Information of the Compound and Protein
Compound Name
1-[[2-(3-chlorophenyl)-5-(trifluoromethyl)pyrazol-3-yl]methyl]-3-(2-oxo-1H-quinolin-5-yl)urea
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Canonical SMILES
FC(F)(F)c1cc(CNC(=O)Nc2cccc3[nH]c(=O)ccc23)n(n1)-c1cccc(Cl)c1
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Compound Formula C21H15ClF3N5O2
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 1.71 nM
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