Brief Information of the Compound and Protein
Compound Name
1-(2-oxo-1H-quinolin-5-yl)-3-[[2-phenylmethoxy-6-(trifluoromethyl)pyridin-3-yl]methyl]urea
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Canonical SMILES
FC(F)(F)c1ccc(CNC(=O)Nc2cccc3[nH]c(=O)ccc23)c(OCc2ccccc2)n1
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Compound Formula C24H19F3N4O3
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 1.2 nM
   TI
   LI
   LO
   TS