Brief Information of the Compound and Protein
Compound Name
(6-fluoro-1-methylbenzimidazol-2-yl)-(7-fluoro-1-methylindol-3-yl)methanone
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Canonical SMILES
Cn1cc(C(=O)c2nc3ccc(F)cc3n2C)c2cccc(F)c12
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Compound Formula C18H13F2N3O
Compound Structure
Protein Name
Proprotein convertase subtilisin/kexin type 9
Protein Classification
Enzyme
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Protease
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Serine protease
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Serine protease SB clan
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Serine protease S8A subfamily
Uniprot ID
Q8NBP7
Gene Name
PCSK9
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000063 Hep-G2 Homo sapiens (Human)  1
1
EC50 = 1.21 nM
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