Brief Information of the Compound and Protein
Compound Name
trans-3-(4-(2,4-difluorobenzyl)piperazin-l-yl)-N-(3-fluorocyclobutyl)-7-methylpyrido[3,4-b]pyrazin-2-amine
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Canonical SMILES
Cc1cc2nc(N[C@H]3C[C@H](F)C3)c(N3CCN(Cc4ccc(F)cc4F)CC3)nc2cn1
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Compound Formula C23H25F3N6
Compound Structure
Protein Name
G-protein coupled receptor 6
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
Uniprot ID
P46095
Gene Name
GPR6
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 49.4 nM
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