Brief Information of the Compound and Protein
Compound Name
1-(1H-indazol-4-yl)-3-[[5-(trifluoromethyl)-2-[4-(trifluoromethyl)phenyl]pyrazol-3-yl]methyl]urea
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Canonical SMILES
FC(F)(F)c1cc(CNC(=O)Nc2cccc3[nH]ncc23)n(n1)-c1ccc(cc1)C(F)(F)F
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Compound Formula C20H14F6N6O
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
Ki = 3.8 nM
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   LI
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