Brief Information of the Compound and Protein
Compound Name
 Compound Info 
1-[2-(cyclopropylmethoxy)ethyl]-3-[5-[2-(5,6-dimethoxypyridin-3-yl)ethynyl]-4-methyl-1,3-thiazol-2-yl]urea
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 PubChem ID
CID: 59615740
Canonical SMILES
COc1cc(cnc1OC)C#Cc1sc(NC(=O)NCCOCC2CC2)nc1C
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Compound Formula C20H24N4O4S
Compound Structure
Protein Name
 Protein Info 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Protein Classification
Enzyme
>
Transferase
Uniprot ID
P48736
Gene Name
PIK3CG
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000040 THP-1
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 180 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 3 nM