Brief Information of the Compound and Protein
Compound Name
 Compound Info 
CAMIZESTRANT
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 PubChem ID
CID: 134453496
Canonical SMILES
C[C@@H]1Cc2c(ccc3[nH]ncc23)[C@@H](c2ccc(NC3CN(CCCF)C3)cn2)N1CC(F)(F)F
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Compound Formula C24H28F4N6
Compound Structure
Protein Name
 Protein Info 
Estrogen receptor
Protein Classification
Transcription factor
>
Nuclear receptor
>
Nuclear hormone receptor subfamily 3
>
Nuclear hormone receptor subfamily 3 group A
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Nuclear hormone receptor subfamily 3 group A member 1
Uniprot ID
P03372
Gene Name
ESR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000083 MCF-7
 Cell Line Info 
Homo sapiens (Human)  4
1
IC50 = 0.1259 nM
   TI
   LI
   LO
   TS
2
IC50 = 0.1585 nM
   TI
   LI
   LO
   TS
3
IC50 = 6.31 nM
   TI
   LI
   LO
   TS
4
IC50 > 316.23 nM
   TI
   LI
   LO
   TS