Brief Information of the Compound and Protein
Compound Name
5-(2-cyclopropylethynyl)-2-(4,4-difluoropiperidin-1-yl)-6-methyl-N-(2-sulfamoylpyridin-4-yl)pyridine-3-carboxamide
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PubChem ID
CID: 146525819
Canonical SMILES
Cc1nc(N2CCC(F)(F)CC2)c(cc1C#CC1CC1)C(=O)Nc1ccnc(c1)S(N)(=O)=O
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Compound Formula C22H23F2N5O3S
Compound Structure
Protein Name
Sodium channel protein type 10 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q9Y5Y9
Gene Name
SCN10A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 12 nM
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