Brief Information of the Compound and Protein
Compound Name
 Compound Info 
US9067937, 28
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 PubChem ID
SID: 163542035
Canonical SMILES
CN(C)C[C@H]1CC[C@@H](CC1)Nc1c(cnc2ccc(nc12)-c1cc(Cl)c(O)c(Cl)c1)C(C)=O
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Compound Formula C25H28Cl2N4O2
Compound Structure
Protein Name
 Protein Info 
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
CMGC protein kinase group
>
CMGC protein kinase DYRK family
>
CMGC protein kinase Dyrk1 subfamily
Uniprot ID
Q13627
Gene Name
DYRK1A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 5 nM
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