Brief Information of the Compound and Protein
Compound Name
(3Z,6R,11aS)-7,8,10-trimethoxy-9-methyl-6-phenyl-3-[(2,4,5-trimethoxy-3-methylphenyl)methylidene]-11,11a-dihydro-6H-pyrazino[1,2-b]isoquinoline-1,4-dione
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PubChem ID
CID: 132942893
Canonical SMILES
COc1cc(\C=C2/NC(=O)[C@@H]3Cc4c(OC)c(C)c(OC)c(OC)c4[C@H](N3C2=O)c2ccccc2)c(OC)c(C)c1OC
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Compound Formula C33H36N2O8
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 4
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9ERZ8
Gene Name
TRPV4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 > 100000 nM
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