Brief Information of the Compound and Protein
Compound Name
5-bromo-4-[4-[(2-methylphenyl)methyl]piperazin-1-yl]-1H-pyridazin-6-one
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PubChem ID
CID: 17466271
Canonical SMILES
Cc1ccccc1CN1CCN(CC1)c1cn[nH]c(=O)c1Br
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Compound Formula C16H19BrN4O
Compound Structure
Protein Name
Short transient receptor potential channel 5
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9UL62
Gene Name
TRPC5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  4
1
IC50 = 4000 nM
   TI
   LI
   LO
   TS
2
IC50 = 4400 nM
   TI
   LI
   LO
   TS
3
IC50 = 5000 nM
   TI
   LI
   LO
   TS
4
IC50 = 7800 nM
   TI
   LI
   LO
   TS