Brief Information of the Compound and Protein
Compound Name
 Compound Info 
N-(2-acetamidoethyl)-N-benzyl-8-butan-2-yl-1-methyl-4H-chromeno[4,3-c]pyrazole-3-carboxamide
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 PubChem ID
CID: 122657507
Canonical SMILES
CCC(C)c1ccc2OCc3c(nn(C)c3-c2c1)C(=O)N(CCNC(C)=O)Cc1ccccc1
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Compound Formula C27H32N4O3
Compound Structure
Protein Name
 Protein Info 
Bile acid receptor
Protein Classification
Transcription factor
>
Nuclear receptor
>
Nuclear hormone receptor subfamily 1
>
Nuclear hormone receptor subfamily 1 group H
>
Nuclear hormone receptor subfamily 1 group H member 4
Uniprot ID
Q96RI1
Gene Name
NR1H4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 23 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 27 nM