Brief Information of the Compound and Protein
Compound Name
6-fluoro-2-(4-methylpiperazin-1-yl)-3-[4-(trifluoromethoxy)phenyl]quinazolin-4-one
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PubChem ID
CID: 155566379
Canonical SMILES
CN1CCN(CC1)c1nc2ccc(F)cc2c(=O)n1-c1ccc(OC(F)(F)F)cc1
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Compound Formula C20H18F4N4O2
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 4
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9HBA0
Gene Name
TRPV4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 2060 nM
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