Brief Information of the Compound and Protein
Compound Name
N-[4-cyclobutyl-5-(2-piperidin-1-ylethyl)-1,3-thiazol-2-yl]-1-(5-fluoropyridin-2-yl)-5-methylpyrazole-4-carboxamide;dihydrochloride
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PubChem ID
CID: 155564707
Canonical SMILES
Cl.Cl.Cc1c(cnn1-c1ccc(F)cn1)C(=O)Nc1nc(C2CCC2)c(CCN2CCCCC2)s1
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Compound Formula C24H31Cl2FN6OS
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 4
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9ERZ8
Gene Name
TRPV4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 0.32 nM
   TI
   LI
   LO
   TS