Brief Information of the Compound and Protein
Compound Name
N-[4-cyclobutyl-5-(4-methylpiperazin-1-yl)-1,3-thiazol-2-yl]-1,5-dimethylpyrazole-4-carboxamide;dihydrochloride
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PubChem ID
CID: 155546887
Canonical SMILES
Cl.Cl.CN1CCN(CC1)c1sc(NC(=O)c2cnn(C)c2C)nc1C1CCC1
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Compound Formula C18H28Cl2N6OS
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 4
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9HBA0
Gene Name
TRPV4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 730 nM
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