Brief Information of the Compound and Protein
Compound Name
 Compound Info 
6-acetyl-2-methoxy-N-[1-[[2-(trifluoromethoxy)phenyl]methyl]-2,3-dihydroindol-5-yl]-7,8-dihydro-5H-1,6-naphthyridine-5-carboxamide
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 PubChem ID
CID: 155530658
Canonical SMILES
COc1ccc2C(N(CCc2n1)C(C)=O)C(=O)Nc1ccc2N(Cc3ccccc3OC(F)(F)F)CCc2c1
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Compound Formula C28H27F3N4O4
Compound Structure
Protein Name
 Protein Info 
Nuclear receptor ROR-gamma
Protein Classification
Transcription factor
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Nuclear receptor
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Nuclear hormone receptor subfamily 1
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Nuclear hormone receptor subfamily 1 group F
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Nuclear hormone receptor subfamily 1 group F member 3
Uniprot ID
P51449
Gene Name
RORC
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000001 Jurkat
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 2000 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 11 nM
2 IC50 = 20 nM