Brief Information of the Compound and Protein
Compound Name
8-Chloro-11-(1-methylpiperidin-4-ylidene)-6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridine fumarate
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PubChem ID
CID: 155555597
Canonical SMILES
CN1CCC(=C2c3ccc(Cl)cc3CCc3cccnc32)CC1.O=C(O)/C=C/C(=O)O
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Compound Formula C24H25ClN2O4
Compound Structure
Protein Name
Histamine H1 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
P35367
Gene Name
HRH1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
Ki = 0.3981 nM
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