Brief Information of the Compound and Protein
Compound Name
13-chloro-2-[1-[(6-methylpyridin-3-yl)methyl]piperidin-4-ylidene]-4-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaene
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PubChem ID
CID: 10070478
SID: 15055826
Canonical SMILES
Cc1ccc(CN2CCC(CC2)=C2c3ccc(Cl)cc3CCc3cccnc23)cn1
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Compound Formula C26H26ClN3
Compound Structure
Protein Name
Histamine H1 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
P35367
Gene Name
HRH1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
Ki = 7.586 nM
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   LI
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