Brief Information of the Compound and Protein
| Compound Name |
Faridak
Show/Hide
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PubChem ID | |||||
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Compound Structure |
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| Protein Name |
Histone deacetylase 3
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Protein Classification |
Epigenetic regulator
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Eraser
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Histone deacetylase
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HDAC class I
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| Uniprot ID | Gene Name | HDAC3 |
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Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
| Cell Line ID | Cell Line Name | Cell Line Organism | |
| CL000023 | BTI-Tn-5B1-4 | Trichoplusia ni (Cabbage looper) | 1 |
| 1 |
IC50 = 5.83 nM
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TI
LI
LO
TS
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|---|---|---|---|
| CL000006 | HEK293 | Homo sapiens (Human) | 1 |
| 1 |
IC50 = 2.1 nM
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TI
LI
LO
TS
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Biochemical Assays
| 1 | IC50 = 1.5 nM | ||
|---|---|---|---|
| 2 | IC50 = 2 nM | ||
| 3 | IC50 = 2.1 nM | ||
| 4 | IC50 < 15 nM | ||
| 5 | IC50 = 15 nM | ||
| 6 | IC50 = 60 nM | ||
| 7 | IC50 < 300 nM | ||
| 8 | Ki = 1.1 nM | ||
| 9 | Ki = 2.3 nM | ||
| 10 | Ki = 2.4 nM | ||