Brief Information of the Compound and Protein
Compound Name
6-methyl-N-[7-methyl-8-[[(3S)-3-methyl-4-(2-methylpropanoyl)piperazin-1-yl]methyl]-[1,2,4]triazolo[1,5-a]pyridin-6-yl]pyridine-3-carboxamide
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PubChem ID
CID: 155536039
Canonical SMILES
CC(C)C(=O)N1CCN(Cc2c(C)c(NC(=O)c3ccc(C)nc3)cn3ncnc23)C[C@@H]1C
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Compound Formula C24H31N7O2
Compound Structure
Protein Name
Nuclear receptor ROR-gamma
Protein Classification
Transcription factor
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Nuclear receptor
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Nuclear hormone receptor subfamily 1
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Nuclear hormone receptor subfamily 1 group F
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Nuclear hormone receptor subfamily 1 group F member 3
Uniprot ID
P51449
Gene Name
RORC
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
IC50 = 230 nM
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