Brief Information of the Compound and Protein
Compound Name
14,15-diazatetracyclo[7.6.1.0^{2,7}.0^{13,16}]hexadeca-1(15),2(7),3,5,9(16),10,12-heptaen-8-one
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PubChem ID
CID: 8515
SID: 15172126
Canonical SMILES
O=C1c2ccccc2-c2n[nH]c3cccc1c23
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Compound Formula C14H8N2O
Compound Structure
Protein Name
Mitogen-activated protein kinase 10
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
CMGC protein kinase group
>
CMGC protein kinase MAPK family
>
CMGC protein kinase JNK subfamily
Uniprot ID
P53779
Gene Name
MAPK10
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Kd = 22 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 90 nM
2 IC50 = 90.5 nM