Brief Information of the Compound and Protein
Compound Name
(5S)-5-[3-(difluoromethyl)pyridin-2-yl]-5-methoxy-8-oxospiro[2.5]oct-6-ene-7-carbonitrile
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PubChem ID
CID: 155566325
Canonical SMILES
CO[C@]1(CC2(CC2)C(=O)C(=C1)C#N)c1ncccc1C(F)F
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Compound Formula C16H14F2N2O2
Compound Structure
Protein Name
Kelch-like ECH-associated protein 1
Protein Classification
Unclassified protein
Uniprot ID
Q14145
Gene Name
KEAP1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 14 nM
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