Brief Information of the Compound and Protein
Compound Name
4,7-dimethyl-5-{3-[4-(2-fluorophenyl)piperazin-1-yl]propoxy}coumarin
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PubChem ID
CID: 139187859
Canonical SMILES
Cc1cc(OCCCN2CCN(c3ccccc3F)CC2)c2c(C)cc(=O)oc2c1
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Compound Formula C24H27FN2O3
Compound Structure
Protein Name
5-hydroxytryptamine receptor 2A
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P28223
Gene Name
HTR2A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
Ki = 55 nM
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