Brief Information of the Compound and Protein
Compound Name
4-((1-(3-chloro-4-(trifluoromethoxy)benzoyl)azetidin-3-yloxy)methyl)-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide
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PubChem ID
CID: 145994290
Canonical SMILES
O=C(c1ccc(OC(F)(F)F)c(Cl)c1)N1CC(OCc2ccc(S(=O)(=O)Nc3ncns3)cc2)C1
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Compound Formula C20H16ClF3N4O5S2
Compound Structure
Protein Name
Sodium channel protein type 3 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q9NY46
Gene Name
SCN3A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 237 nM
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