Brief Information of the Compound and Protein
Compound Name
7-[4-(6-methoxypyridin-3-yl)oxypiperidin-1-yl]-6-methyl-1H-pyrido[2,3-d]pyrimidine-2,4-dione
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PubChem ID
CID: 135171475
Canonical SMILES
COc1ccc(OC2CCN(CC2)c2nc3[nH]c(=O)[nH]c(=O)c3cc2C)cn1
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Compound Formula C19H21N5O4
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 18 nM
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