Brief Information of the Compound and Protein
Compound Name
3-methyl-6-methylsulfonyl-2-(4-phenoxypiperidin-1-yl)-5,7-dihydropyrrolo[3,4-b]pyridine
    Show/Hide
PubChem ID
CID: 135150406
Canonical SMILES
Cc1cc2CN(Cc2nc1N1CCC(CC1)Oc1ccccc1)S(C)(=O)=O
    Show/Hide
Compound Formula C20H25N3O3S
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Monoamine receptor
>
Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 20 nM
   TI
   LI
   LO
   TS