Brief Information of the Compound and Protein
Compound Name
[4-chloro-6-[(3S,4R)-3-fluoro-4-(1H-indazol-5-yloxy)piperidin-1-yl]-5-methylpyrimidin-2-yl]methanol
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PubChem ID
CID: 135150478
Canonical SMILES
Cc1c(Cl)nc(CO)nc1N1CC[C@@H](Oc2ccc3[nH]ncc3c2)[C@@H](F)C1
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Compound Formula C18H19ClFN5O2
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 20 nM
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